Solid phase synthesis of 2-substituted benzofurans via the palladium-catalysed heteroannulation of acetylenes

Daniele Fancelli; Maria Chiara Fagnola; Dino Severino; Angelo Bedeschi

doi:10.1016/S0040-4039(97)00301-8

Solid phase synthesis of 2-substituted benzofurans via the palladium-catalysed heteroannulation of acetylenes

Daniele Fancelli, Maria Chiara Fagnola, Dino Severino, Angelo Bedeschi

Istituto Europeo di Oncologia

Research output: Contribution to journal › Article › peer-review

Abstract

The copper/palladium-promoted heterannulation of terminal acetylenic compounds in the presence of resin bound ortho-hydroxy aryl iodides is described. The process produces 2-substituted benzofuran derivatives in good yield and high purity.

Original language	English
Pages (from-to)	2311-2314
Number of pages	4
Journal	Tetrahedron Letters
Volume	38
Issue number	13
DOIs	https://doi.org/10.1016/S0040-4039(97)00301-8
Publication status	Published - Mar 31 1997

ASJC Scopus subject areas

Biochemistry
Organic Chemistry
Drug Discovery

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title = "Solid phase synthesis of 2-substituted benzofurans via the palladium-catalysed heteroannulation of acetylenes",

abstract = "The copper/palladium-promoted heterannulation of terminal acetylenic compounds in the presence of resin bound ortho-hydroxy aryl iodides is described. The process produces 2-substituted benzofuran derivatives in good yield and high purity.",

author = "Daniele Fancelli and Fagnola, {Maria Chiara} and Dino Severino and Angelo Bedeschi",

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T1 - Solid phase synthesis of 2-substituted benzofurans via the palladium-catalysed heteroannulation of acetylenes

AU - Fancelli, Daniele

AU - Fagnola, Maria Chiara

AU - Severino, Dino

AU - Bedeschi, Angelo

PY - 1997/3/31

Y1 - 1997/3/31

N2 - The copper/palladium-promoted heterannulation of terminal acetylenic compounds in the presence of resin bound ortho-hydroxy aryl iodides is described. The process produces 2-substituted benzofuran derivatives in good yield and high purity.

AB - The copper/palladium-promoted heterannulation of terminal acetylenic compounds in the presence of resin bound ortho-hydroxy aryl iodides is described. The process produces 2-substituted benzofuran derivatives in good yield and high purity.

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JO - Tetrahedron Letters

JF - Tetrahedron Letters

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